R.M. Versteegen, W. ten Hoeve, R. Rossin M.A.R. de Geus, H.M. Janssen, M.S. Robillard; Click‐to‐Release from trans‐Cyclooctenes: Mechanistic Insights and Expansion of Scope from Established Carbamate to Remarkable Ether Cleavage, Angew. Chem. Int. Ed. 2018, published online 10 May 2018. doi: 10.1002/anie.201800402

R. Rossin, R.M. Versteegen, J. Wu, A. Khasanov, H.J. Wessels, E.J. Steenbergen, W. ten Hoeve, H.M. Janssen, A.H.A.M. van Onzen, P.J. Hudson, M.S. Robillard; Chemically triggered drug release from an antibody-drug conjugate leads to potent antitumour activity in mice, Nat.Comm. 2018, 9, 1484. doi:10.1038/s41467-018-03880-y

R. Rossin, S.M.J. van Duijnhoven, W. ten Hoeve, H.M. Janssen, L.H.J. Kleijn, F.J.M. Hoeben, R.M. Versteegen, M.S. Robillard; Triggered drug release from an antibody-drug conjugate  using fast “Click-to-release” chemistry in mice. Bioconj.Chem., 2016 27(7):1697-1706.  doi:10.1021/acs.bioconjchem.6b00231

S. van Duijnhoven, R. Rossin, S. van den Bosch, M. Wheatcroft, P. Hudson, M. Robillard; CC49 diabody pretargeting using click chemistry in vivo. J.Nucl.Med. 2015, 54, 1989–1995. doi:10.2967/jnumed.115.159145

R. Rossin and M.S. Robillard; Pretargeted imaging using bioorthogonal chemistry in mice. Current Opinion in Chemical Biology 2014, 21:161-169. doi/10.1016/j.cbpa.2014.07.023

R. Rossin, S.M.J. van Duijnhoven, T. Läppchen, S.M. van den Bosch, M.S. Robillard; Trans-cyclooctene tag with improved properties for tumor pretargeting with the Diels-Alder reaction. Mol. Pharmaceutics 2014, 11(9), 3090-3096. doi:10.1021/mp500275a

R.M. Versteegen, R. Rossin, W. ten Hoeve, H.M. Janssen, M.S. Robillard; Click to release: Instantaneous doxorubicin elimination upon tetrazine ligation. Angew. Chem. Int. Ed. 2013, 52, 14112–14116. doi:10.1002/anie.201305969

R. Rossin, T. Läppchen, S.M. van den Bosch, R. Laforest, M.S. Robillard; Diels-Alder reaction for tumor pretargeting: In vivo chemistry can boost tumor radiation dose compared with directly labeled antibody. J. Nucl. Med. 2013, 54, 11, 1989-1995. doi:10.2967/jnumed.113.12.3745

R. Rossin, S.M. van den Bosch, W. ten Hoeve, M. Carvelli, R.M. Versteegen, J. Lub, M.S. Robillard; Highly reactive trans-cyclooctene tags with improved stability for Diels-Alder chemistry in living systems. Bioconjug. Chem. 2013, 24, 7, 1210–1217. doi:10.1021/bc400153y

S.M. van den Bosch, R. Rossin, P. Renart Verkerk, W. ten Hoeve, H.M. Janssen, J. Lub, M.S. Robillard; Evaluation of strained alkynes for Cu-free click reaction in live mice. Nucl. Med. Biol. 2013, 40, 415-423. doi: 10.1016/j.nucmedbio.2012.12.006  

D.J. Vugts, A. Vervoort, M. Stigter-van Walsum, G.W.M. Visser, M.S. Robillard, R.M. Versteegen, R.C.M. Vulders, J.D.M. Herscheid, G.A.M.S. van Dongen; Synthesis of Phosphine and Antibody–Azide Probes for in Vivo Staudinger Ligation in a Pretargeted Imaging and Therapy Approach. Bioconjug. Chem. 2011, 22, 10, 2072–2081. doi: 10.1021/bc200298v

R. Rossin, P. Renart Verkerk, S.M. van den Bosch, R.C.M. Vulders, I. Verel, J. Lub, M.S. Robillard; In Vivo Chemistry for Pretargeted Tumor Imaging in Live Mice. Angew. Chem. Int. Ed. 2010, 49, 3375-3378. doi: 10.1002/anie.200906294; featured in Nature Nanotechnology 2010, 5, 384. doi:10.1038/nnano.2010.122

R. van Brakel, R.C.M. Vulders, R.J. Bokdam, H. Grüll, M.S. Robillard; A Doxorubicin Prodrug Activated by the Staudinger Reaction. Bioconjugate Chem. 2008, 19, 3, 714-718. doi: 10.1021/bc700394s